e.g. Filippa Pettersson or Cancer Res. 75(6) , 1102-12, (2015) or 10.1002/anie.201600521
Gold-catalysed cascade rearrangements of ynamide propargyl esters
SJ Heffernan, JM Beddoes, MF Mahon…
Index: Heffernan, Stephen J.; Beddoes, James M.; Mahon, Mary F.; Hennessy, Alan J.; Carbery, David R. Chemical Communications, 2013 , vol. 49, # 23 p. 2314 - 2316
The Au (I)-catalysed rearrangement of propargylic esters formed from an ynamide has been studied. The reaction is facile, and when conducted in the presence of a reactive indole nucleophile, leads to a cascade process whereby γ-indolyl α-acyloxyenamides are formed ...