Efficient nickel-mediated intramolecular amination of aryl chlorides

R Omar-Amrani, A Thomas, E Brenner…

Index: Kiguchi, Toshiko; Kuninobu, Naoko; Takahashi, Yoshiko; Yoshida, Yukiyo; Naito, Takeaki; Ninomiya, Ichiya Synthesis, 1989 , # 10 p. 778 - 781

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Citation Number: 137

Abstract

... provide access to the desired ring system (Pd(PPh 3 ) 4 (10 mol %), NaO-t ... The complexes show good catalytic activity for the synthesis of indoles, quinolines, benzazepines ... Intramolecular palladium-catalyzed aryl amination and aryl amidation. Wolfe, John P.; Rennels, Roger A ...

~7%

~39%

~3%

~69%

~62%

~11%

~90%

Nitrogen Assistance in Intramolecular Nickel-Promoted Tandem...

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Facile Synthesis of 2-Benzylindoles

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Enantioselective TADMAP-catalyzed carboxyl migration reactio...

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