PF-04859989 as a template for structure-based drug design: Identification of new pyrazole series of irreversible KAT II inhibitors with improved lipophilic efficiency

AB Dounay, M Anderson, BM Bechle, E Evrard…

Index: Bioorganic and Medicinal Chemistry Letters, , vol. 23, # 7 p. 1961 - 1966

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Citation Number: 13

Abstract

... Bioorganic & Medicinal Chemistry Letters. Volume 23, Issue 7, 1 April 2013, Pages 1961–1966. Cover image Cover image. ... Research and Development, Neuroscience Medicinal Chemistry, Groton Laboratories, Eastern Point Road, Groton, CT 06340, United States. ...

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