Synthesis of one??, two??and three??ring macrocyclic, bifunctional compounds for use in radiolabelling monoclonal antibodies

…, LF Lindoy, SV Smith, JG Wilson

Index: Ramli, Martalena; Dong, Ying; Lindoy, Leonard F.; Smith, Suzanne V.; Wilson, J. Gerald Journal of Heterocyclic Chemistry, 2005 , vol. 42, # 1 p. 77 - 83

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Citation Number: 4

Abstract

Abstract The synthesis of new linked bis-and tris-ring tetraazamacrocyclic (bifunctional) reagents for use in an alternative strategy for radiolabelling antibodies is described. For comparison with the above systems, a new single ring bifunctional system incorporating a dioxocyclam ring is also reported.