Optimization of Triazine Nitriles as Rhodesain Inhibitors: Structure–Activity Relationships, Bioisosteric Imidazopyridine Nitriles, and X??ray Crystal Structure Analysis …

V Ehmke, E Winkler, DW Banner, W Haap…

Index: ChemMedChem, , vol. 8, # 6 p. 967 - 975

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Citation Number: 7

Abstract

... Nitriles as Rhodesain Inhibitors: Structure–Activity Relationships, Bioisosteric Imidazopyridine Nitriles, and X-ray Crystal Structure Analysis with Human Cathepsin L. ChemMedChem, 8: 967–975. ... Volume: Issue: Page: ... Thumbnail image of. 16a, Thumbnail image of. 4.16, 8, 33. ...

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Optimization of Triazine Nitriles as Rhodesain Inhibitors: S...

[Ehmke, Veronika; Winkler, Edwin; Banner, David W.; Haap, Wolfgang; Schweizer, W. Bernd; Rottmann, Matthias; Kaiser, Marcel; Freymond, Celine; Schirmeister, Tanja; Diederich, Francois ChemMedChem, 2013 , vol. 8, # 6 p. 967 - 975]