Design and synthesis of conformationally constrained inhibitors of non-nucleoside reverse transcriptase

…, P Felock, V Munshi, D DiStefano, J Flynn…

Index: Grzegozek, Maria Journal of Heterocyclic Chemistry, 2008 , vol. 45, # 6 p. 1879 - 1882

Full Text: HTML

Citation Number: 18

Abstract

... Journal ... J. Med. Chem. ... Phone: 215-652-4715. Fax: 215-652-3971. E-mail: Robert_gomez@merck. com. ● Author Present Address. Department of Boston Discovery Chemistry, Merck Research Labs., 33 Avenue Louis Pasteur, Boston, Massachusetts 02115-5717, United States. ...

~92%

~60%

~69%

1H-imidazo [4, 5-c] quinolin-4-amines: novel non-xanthine ad...

[Galen, Philip J. M. van; Nissen, Peter; Wijngaarden, Ineke van; IJzerman, Adriaan P.; Soudijn, Willem Journal of Medicinal Chemistry, 1991 , vol. 34, # 3 p. 1202 - 1206]

The Synthesis of Some 3-Nitro-and 3-Amino-4-dialkylaminoalky...

[Surrey; Cutler Journal of the American Chemical Society, 1951 , vol. 73, p. 2413,2414]

Substituted terphenyl compounds as the first class of low mo...

[Goeblyoes, Aniko; Gao, Zhan-Guo; Brussee, Johannes; Connestari, Roberto; Santiago, Sabrina Neves; Ye, Kai; Ijzerman, Adriaan P.; Jacobson, Kenneth A. Journal of Medicinal Chemistry, 2006 , vol. 49, # 11 p. 3354 - 3361]