Tetrahedron

Synthesis and reactivity of 2-(1', 3'dithian-2'-yl) indoles

M Rubiralta, N Casamitjana, DS Grierson, HP Husson

Index: Rubiralta, Mario; Casamitjana, Nuria; Grierson, David S.; Husson, Henri-Philippe Tetrahedron, 1988 , vol. 44, # 2 p. 443 - 450

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Citation Number: 17

Abstract

The 2-(1', 3'-dithian-2'-yl) indoles 1 a, b were prepared in a single operation involving reaction of the onions of the N-protected indoles 3 a, b with 2-chloro-1, 3-dithiane. Subsequent reaction of 1 a with excess n-BuLi followed by an electrophile (1-methyl-4- ...