1-(2-Hydroxy-2-methyl-3-phenoxypropanoyl) indoline-4-carbonitrile derivatives as potent and tissue selective androgen receptor modulators

ELP Chekler, R Unwalla, TA Khan…

Index: Journal of Medicinal Chemistry, , vol. 57, # 6 p. 2462 - 2471

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Citation Number: 3

Abstract

... Journal of Medicinal ... BioTherapeutics Medicinal Chemistry, Pfizer Global Research and Development, 200 Cambridgepark Drive, Cambridge, Massachusetts 02140, United States. ... The pharmaceutical industry has been exploring the use of agents that selectively activate AR ...

1-(2-Hydroxy-2-methyl-3-phenoxypropanoyl) indoline-4-carboni...

[Chekler, Eugene L. Piatnitski; Unwalla, Rayomond; Khan, Taukeer A.; Tangirala, Raghuram S.; Johnson, Mark; St. Andre, Michael; Anderson, James T.; Kenney, Thomas; Chiparri, Sue; McNally, Chris; Kilbourne, Edward; Thompson, Catherine; Nagpal, Sunil; Weber, Gregory; Schelling, Scott; Owens, Jane; Morris, Carl A.; Powell, Dennis; Verhoest, Patrick R.; Gilbert, Adam M. Journal of Medicinal Chemistry, 2014 , vol. 57, # 6 p. 2462 - 2471]

Regioselective cyanation of 3-substituted pyridine 1-oxides

[Heterocycles, , vol. 22, # 1 p. 93 - 96]