An Efficient Synthesis of 3-Substituted N-Glycoside Indoles Useful as Sodium-Dependent Glucose Transporter Inhibitors

X Li, KM Wells, S Branum, S Damon…

Index: Organic Process Research and Development, , vol. 16, # 11 p. 1727 - 1732

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Abstract

... Organic Process Research & Development. ... Cyclopropylaryl Bromide and Subsequent Grignard Formation Process Development Since aryl bromide 8 was not commercially available in ... The discovery route followed the procedure outlined by Himmelsbach et al., which gave four ...