Tetrahedron letters

Preparation of 6-chloro-5-fluoroindole via the use of palladium and copper-mediated heterocyclisations

DR Adams, MAJ Duncton, JRA Roffey, J Spencer

Index: Adams, David R.; Duncton, Matthew A.J.; Roffey, Jonathan R.A.; Spencer, John Tetrahedron Letters, 2002 , vol. 43, # 42 p. 7581 - 7583

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Citation Number: 24

Abstract

Download PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... The title indole, the heterocyclic core of the 5-HT 2C receptor agonist Ro 60-0175, was prepared by a modification to the Stille indole synthesis, or by the method of Gonzalez and co-workers. ... The title indole was prepared by either stoichiometric copper- or catalytic palladium-mediated ...