Synthesis and Biological Properties of Enkephalin??like Peptides Containing Carboranylalanine in Place of Phenylalanine

R Schwyzer, KQ Do, AN Eberle…

Index: Schwyzer; Do; Eberle; Fauchere Helvetica Chimica Acta, 1981 , vol. 64, # 7 p. 2078 - 2083

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Citation Number: 27

Abstract

Abstract The syntheses of [D-Ala 2, Car 4, Leu 5]-enkephalin, its amide, and of [D-Ala 2, Car 4, Met 5]-enkephalin amide are described in detail. The three compounds show pronounced morphine-like potencies in certain bio-assays, and were used to investigate the influence of

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Synthesis of chiral α-amino acids

[Chakraborty, Tushar K.; Ghosh, Animesh Tetrahedron Letters, 2002 , vol. 43, # 52 p. 9691 - 9693]