Structure guided optimization of a fragment hit to imidazopyridine inhibitors of PI3K

S Pecchi, ZJ Ni, W Han, A Smith, J Lan…

Index: Bioorganic and Medicinal Chemistry Letters, , vol. 23, # 16 p. 4652 - 4656

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Abstract

... Please enable JavaScript to use all the features on this page. Bioorganic & Medicinal Chemistry Letters. Volume 23, Issue 16, 15 August 2013, Pages 4652–4656. Cover image Cover image. ... Chemistry, Novartis Institutes for Biomedical Research, Emeryville, CA, USA; ...