Synthesis and in vitro evaluation of N-substituted maleimide derivatives as selective monoglyceride lipase inhibitors

N Matuszak, GG Muccioli, G Labar…

Index: Journal of Medicinal Chemistry, , vol. 52, # 23 p. 7410 - 7420

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Citation Number: 78

Abstract

... Journal of Medicinal ... 2009, 52 (23), pp 7410–7420. DOI: 10.1021/jm900461w. Publication Date (Web): July 7, 2009. Copyright © 2009 American Chemical Society. ... From a medicinal chemistry point of view, few MGL inhibitors are available and they often lack selectivity or have not ...