Organic Process Research & Development

Practical amination of nitropyridones by silylation

RA Singer, M Doré

Index: Organic Process Research and Development, , vol. 12, # 6 p. 1261 - 1264

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Citation Number: 5

Abstract

... 3-nitro-4-pyridone (1) was coupled with various primary amines in a tandem process (Table 2 ... General Procedure for Amination of Nitropyridones To a suspension of the nitropyridone (5.00 g, 35.7 ... and once with a saturated aqueous solution of NaCl (33 L). The organic layer was ...