Tetrahedron

A general and efficient PIFA mediated synthesis of heterocycle-fused quinolinone derivatives

MT Herrero, I Tellitu, E Domı́nguez, S Hernández…

Index: Herrero, M.Teresa; Tellitu, Imanol; Dominguez, Esther; Hernandez, Susana; Moreno, Isabel; SanMartin, Raul Tetrahedron, 2002 , vol. 58, # 42 p. 8581 - 8589

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Citation Number: 45

Abstract

A new application of the hypervalent iodine reagent phenyliodine (III) bis (trifluoroacetate)(PIFA) has been developed for the construction of a series of N, O, S- containing heterocycle-fused quinolinone derivatives in a general and efficient way. An alternative approach to the formation of these novel tricyclic heterocycles by a PIFA mediated aryl–heteroaryl coupling reaction is also presented.