Design, synthesis, and insecticidal activity of novel pyrazole derivatives containing α-hydroxymethyl-N-benzyl carboxamide, α-chloromethyl-N-benzyl carboxamide, …

…, Y Liu, L Xiong, Y Li, N Yang, Q Wang

Index: Song, Hongjian; Liu, Yuxiu; Xiong, Lixia; Li, Yongqiang; Yang, Na; Wang, Qingmin Journal of Agricultural and Food Chemistry, 2012 , vol. 60, # 6 p. 1470 - 1479

Full Text: HTML

Citation Number: 35

Abstract

On the basis of commercial insecticides tebufenpyrad and tolfenpyrad, two series of novel pyrazole-5-carboxamides containing α-hydroxymethyl-N-benzyl or α-chloromethyl-N-benzyl and pyrazoles containing 4, 5-dihydrooxazole moieties were designed and synthesized via the key intermediate 2-amino-1-(4-substituted) phenyl ethanol. The structures of target compounds were confirmed by 1H NMR and elemental analysis or high-resolution mass ...