Phenethylthiazolethiourea (PETT) compounds, a new class of HIV-1 reverse transcriptase inhibitors. 1. Synthesis and basic structure-activity relationship studies of …

FW Bell, AS Cantrell, M Hoegberg…

Index: Journal of Medicinal Chemistry, , vol. 38, # 25 p. 4929 - 4936

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Citation Number: 421

Abstract

... LY73497 (1) ED,, 1.3 1M 1 2 3 4 IC,, 0.9 )IM 0 1995 American Chemical Society Page 2. 4930 Journal of Medicinal Chemistry, 1995, Vol. 38, No. 25 Table 1. Inhibition of HIV-1: Modification of Quadrant 1 s 3 R~NJ$+N H H Bell et al. anti-HIV-1 activity ...