An efficient synthesis of raloxifene in ionic liquid: a green approach

…, AS Renge, GH Patil, AB Rode, RR Pawar

Index: Shinde, Pravin S.; Shinde, Sandip S.; Renge, Atul S.; Patil, Gajanan H.; Rode, Ambadas B.; Pawar, Rajendra R. Letters in Organic Chemistry, 2009 , vol. 6, # 1 p. 8 - 10

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Citation Number: 17

Abstract

Abstract: An efficient and green procedure for the synthesis of raloxifene has been developed by using Suzuki couplings, Friedel-Crafts acylation, and copper catalyzed coupling reactions in an ionic liquid. Keywords: Raloxifene, ionic liquids, Suzuki coupling, Friedel-Crafts acylation.

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