Reduction of hERG inhibitory activity in the 4-piperidinyl urea series of H3 antagonists

M Berlin, YJ Lee, CW Boyce, Y Wang…

Index: Bioorganic and Medicinal Chemistry Letters, , vol. 20, # 7 p. 2359 - 2364

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Citation Number: 5

Abstract

... Bioorganic & Medicinal Chemistry Letters. ... Chemical Research, Cardiovascular/ Metabolic Diseases and CNS Discovery, and Drug Metabolism and Pharmacokinetics, Merck Research Laboratories, Kenilworth, NJ 07033, USA. ...