Tetrahedron Letters

The aza-robinson annulation: An application to the synthesis of iso-A58365A

FG Fang, M Prato, G Kim, SJ Danishefsky

Index: Fang, Francis G.; Prato, Maurizio; Kim, Guncheol; Danishefsky, Samuel J. Tetrahedron Letters, 1989 , vol. 30, # 28 p. 3625 - 3628

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Citation Number: 58

Abstract

Download full text in PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... Annulation of diazomethylvinylketone (4a) with a variety of secondary thiolactams provides a novel route to dihydro-γ-pyridones. This approach has been applied to the synthesis of iso-A58365A (2), the γ-pyridone analog of the ACE inhibitor, A58365A (1).

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