e.g. Filippa Pettersson or Cancer Res. 75(6) , 1102-12, (2015) or 10.1002/anie.201600521
Synthesis
Synthesis of substituted 8-methoxyquinolines by regioselective bromine-lithium exchange of 5, 7-dihalo-8-methoxyquinolines and 7-bromo-8-methoxyquinoline