Synthesis and optimization of novel (3S, 5R)-5-(2, 2-dimethyl-5-oxo-4-phenylpiperazin-1-yl) piperidine-3-carboxamides as orally active renin inhibitors

Y Mori, Y Ogawa, A Mochizuki, Y Nakamura…

Index: Bioorganic and Medicinal Chemistry, , vol. 21, # 18 p. 5907 - 5922

Full Text: HTML

Citation Number: 5

Abstract

... Bioorganic & Medicinal Chemistry. ... f Medicinal Safety Research Laboratories, Daiichi Sankyo Co., Ltd, 1-16-13 Kitakasai, Edogawa-ku, Tokyo 134-8630, Japan; g Daiichi Sankyo Life Science Research Center in India, Daiichi Sankyo India Pharma Pvt. ... 2. Chemistry. ...