CRTH2 antagonist MK-7246: a synthetic evolution from discovery through development

C Molinaro, PG Bulger, EE Lee, B Kosjek…

Index: Journal of Organic Chemistry, , vol. 77, # 5 p. 2299 - 2309

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Citation Number: 24

Abstract

... Journal of Organic Chemistry. ... J. Org. Chem. , 2012, 77 (5), pp 2299–2309. DOI: 10.1021/jo202620r. Publication Date (Web): February 15, 2012. Copyright © 2012 American Chemical Society. *E-mail: (CM) carmela_molinaro@merck.com, (PGB) paul_bulger@merck.com. ...