Tetrahedron letters

Directed lithiation of N-(tert-butoxycarbonyl) aminoisoxazole: synthesis of 4-substituted aminoisoxazoles

T Konoike, Y Kanda, Y Araki

Index: Konoike, Toshiro; Kanda, Yasuhiko; Araki, Yoshitaka Tetrahedron Letters, 1996 , vol. 37, # 19 p. 3339 - 3342

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Citation Number: 13

Abstract

Download full text in PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... Directed lithiation of 3-(Boc-amino)isoxazole 4 and 5-(Boc-amino)isoxazole 9 is described. Dilithioisoxazoles reacted with a variety of electrophiles to give the corresponding 4-substituted isoxazoles. ... Directed lithiation of 3-Boc-aminoisoxazole and 5-Boc-aminoisoxazole is described.