A new class of potent non-imidazole H 3 antagonists: 2-aminoethylbenzofurans

M Cowart, JK Pratt, AO Stewart, YL Bennani…

Index: Bioorganic and Medicinal Chemistry Letters, , vol. 14, # 3 p. 689 - 693

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Citation Number: 83

Abstract

... Bioorganic & Medicinal Chemistry Letters. Volume 14, Issue 3, 9 February 2004, Pages 689–693. ... However, in spite of the likely medical utility of H 3 antagonists, no agent in the class has yet received clinical approval, perhaps due to inadequate drug-like properties. ...