Tetrahedron letters

An efficient asymmetric synthesis of (R)-3-amino-2, 3, 4, 5-tetrahydro-1H-[1] benzazepin-2-one

JD Armstrong, KK Eng, JL Keller, RM Purick…

Index: Armstrong, Joseph D. III; Eng, Kan K.; Keller, Jennifer L.; Purick, Robert M.; Hartner, Frederick W. Jr.; et al. Tetrahedron Letters, 1994 , vol. 35, # 20 p. 3239 - 3242

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Citation Number: 41

Abstract

Download full text in PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... Two approaches for the asymmetric preparation of (−)- or (+)- α-aminobenzlactam 1 are described. One route is based on the asymmetric hydrogenation of enamide 5 and the other on the racemization/resolution of (±)- 1. ... Two approaches for the asymmetric ...