e.g. Filippa Pettersson or Cancer Res. 75(6) , 1102-12, (2015) or 10.1002/anie.201600521
Concurrent oxygen-18 exchange accompanying the acid-catalyzed hydrolysis of anilides. Implications for the lifetimes of reversibly formed intermediates
AJ Bennet, H Slebocka-Tilk, RS Brown…
Index: Bennet; Slebocka-Tilk; Brown; Guthrie, J. Peter; Jodhan Journal of the American Chemical Society, 1990 , vol. 112, # 23 p. 8497 - 8506
Abstract: Hydrolysis of acetanilide and N, 2, 4-trimethylacetanilide in acid is accompanied by oxygen exchange. The log k,, and log k,, vs-log [H+] profiles are parallel and show no significant divergence. The deuterium solvent kinetic isotope effects on exchange and hydrolysis are unity. A possible alternative mechanism for exchange in acetanilides involving enolization and elimination to give a transient keteniminium ion has been ruled ...