Discovery of ectoparasiticidal hydrazonotrifluoromethanesulfonanilides

…, AG Riches, RM Sargent, DG Sawutz, KA Turner…

Index: Ali, Abdelselam; Fisara, Petr; Freemont, Jamie A.; Kyi, Stella; Meyer, Adam G.; Riches, Andrew G.; Sargent, Roger M.; Sawutz, David G.; Turner, Kathleen A.; Winzenberg, Kevin N.; Yang, Qi Bioorganic and Medicinal Chemistry Letters, 2010 , vol. 20, # 2 p. 649 - 652

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Citation Number: 7

Abstract

... 27, A, D, Me, Me, 3-Cl–Ph, 100, 14.6, 100, 2.6. 28, A, D, Me, Me, 3-F–Ph, 100, 13.4, 100, 2.0. 29, A, D, Me, Et, 3-F–Ph, 100, 7.46, 98, 2.1. 30, G, H, Me, Me, 3-CF 3 –Ph, 98, 95, 0.68. 31, C, A, Me, Me, 2-Cl–Ph, 100, 90, 32, A, D, Me, Et, 2-Cl–Ph, 89, 83, 33, A, D, Me, Me, 2-F–Ph, 100, 8.66, 100, 1.6. ... Reagents and conditions:15 (M) EtOH, 100°C, sealed tube, 16h; (N) EtOH, rt, 16h; ... Reagents and conditions:15 (M) EtOH, 100°C, sealed tube, 16h; (N) EtOH, rt, 16h; ... ...