Optimization of non-ATP competitive CDK/cyclin groove inhibitors through REPLACE-mediated fragment assembly

S Liu, PN Premnath, JK Bolger, TL Perkins…

Index: Journal of Medicinal Chemistry, , vol. 56, # 4 p. 1573 - 1582

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Citation Number: 14

Abstract

... Journal of Medicinal Chemistry. ... Chem. , 2013, 56 (4), pp 1573–1582. DOI: 10.1021/jm3013882. Publication Date (Web): January 16, 2013. Copyright © 2013 American Chemical Society. *E-mail mcinnes@sccp.sc.edu; phone (803) 576-5684. § Author Contributions. ...