Synlett

Traceless solid-phase synthesis of mappicine ketone library via multiple chemoselective palladium-catalyzed reactions on benzenesulfonate linker

H Tsukamoto, R Suzuki, Y Kondo

Index: Synlett, , # 13 p. 2005 - 2010

Full Text: HTML

Citation Number: 2

Abstract

... Synlett 2008(13): 2005-2010 DOI: 10.1055/s ... Commercially available 5-hydroxyanthranilic acid (8) was converted into its methyl ester [8] and the hydroxyl group was selectively tosylated with p-toluenesulfonyl chloride and triethylamine in the presence of an amino group. ...