Optimization of 3, 5-dimethylisoxazole derivatives as potent bromodomain ligands

DS Hewings, O Fedorov…

Index: Journal of Medicinal Chemistry, , vol. 56, # 8 p. 3217 - 3227

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Citation Number: 63

Abstract

... Journal of Medicinal Chemistry. ... Department of Chemistry, Chemistry Research Laboratory, University of Oxford, Mansfield Road, Oxford, OX1 3TA, UK. ‡ Nuffield Department of Clinical Medicine, Structural Genomics Consortium, University of Oxford, Old Road Campus ...