A practical and scalable synthesis of SR 142801, a tachykinin NK3 antagonist

HG Chen, FZ Chung, OP Goel, D Johnson…

Index: Bioorganic and Medicinal Chemistry Letters, , vol. 7, # 5 p. 555 - 560

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Citation Number: 13

Abstract

... Bioorganic & Medicinal Chemistry Letters. Volume 7, Issue 5, 4 March 1997, Pages 555–560. ... The absolute configuration of the key intermediate 7 was determined by single crystal X-ray crystallography, on the basis of which, the absolute configuration of SR 142801 should be (R ...

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