Tetrahedron letters

Concise and regiospecific syntheses of tri-substituted 1, 2, 4-triazoles

…, HP Weber, G Rihs, H Widmer, EK Dziadulewicz

Index: Dunstan, Andrew R.; Weber, Hans-Peter; Rihs, Grety; Widmer, Hans; Dziadulewicz, Edward K. Tetrahedron Letters, 1998 , vol. 39, # 43 p. 7983 - 7986

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Citation Number: 22

Abstract

Download full text in PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... Novel tri-substituted 1,2,4-triazoles are synthesized via complementary, regiospecific routes as part of a lead finding exercise. A key feature of one of the syntheses is recognition of an intrinsic regioselectivity toward deprotonation in the 1-phenylguanazole substrate.