Potent, orally active corticotropin-releasing factor receptor-1 antagonists containing a tricyclic pyrrolopyridine or pyrazolopyridine core

B Dyck, DE Grigoriadis, RS Gross, Z Guo…

Index: Journal of Medicinal Chemistry, , vol. 48, # 12 p. 4100 - 4110

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Citation Number: 24

Abstract

... Journal of Medicinal Chemistry. ... Departments of Medicinal Chemistry, Pharmacology and Lead Discovery, and Preclinical Development, Neurocrine Biosciences, 12790 El Camino Real, San Diego, California 92130. J. Med. Chem. ... Results and Discussion. Chemistry. ...