Large amino acid transporter 1 (LAT1) prodrugs of valproic acid: new prodrug design ideas for central nervous system delivery

L Peura, K Malmioja, K Laine, J Leppänen…

Index: Molecular Pharmaceutics, , vol. 8, # 5 p. 1857 - 1866

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Citation Number: 37

Abstract

... Pharmaceutics , 2011, 8 (5), pp 1857–1866. DOI: 10.1021/mp2001878. Publication Date (Web): July 19 ... small molecular weight drugs and practically none of the large molecular weight drugs ... Consequently, several drug molecules in clinical use such as melfalan,(8) gabapentin,(9 ...