Design, synthesis, and SAR studies of 4-substituted methoxylbenzoyl-aryl-thiazoles analogues as potent and orally bioavailable anticancer agents

Y Lu, CM Li, Z Wang, J Chen, ML Mohler…

Index: Journal of Medicinal Chemistry, , vol. 54, # 13 p. 4678 - 4693

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Citation Number: 44

Abstract

... Journal of Medicinal Chemistry. ... Department of Pharmaceutical Sciences, University of Tennessee, Health Science Center, Memphis, Tennessee 38163, United States. GTx Inc., Preclinical R&D, Memphis, Tennessee 38163, United States. J. Med. Chem. ...

The synthesis and activity of oxazole and thiazole analogues...

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Phenyloxazoles and phenylthiazoles as benzamide bioisosteres...

[Einsiedel, Juergen; Thomas, Christoph; Huebner, Harald; Gmeiner, Peter Bioorganic and Medicinal Chemistry Letters, 2000 , vol. 10, # 17 p. 2041 - 2044]

Phenyloxazoles and phenylthiazoles as benzamide bioisosteres...

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Über 4??Formyl??thiazole

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Synthesis and in??vitro Cytotoxicity of Poly??functionalized...

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