Tetrahedron

Copper-catalyzed synthesis of α, β-unsaturated acylamides via direct amidation from cinnamic acids and N-substituted formamides

H Yan, H Yang, L Lu, D Liu, G Rong, J Mao

Index: Yan, Hong; Yang, Hailong; Lu, Linhua; Liu, Defu; Rong, Guangwei; Mao, Jincheng Tetrahedron, 2013 , vol. 69, # 35 p. 7258 - 7263

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Citation Number: 4

Abstract

Download PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... A highly effective synthesis of α,β-unsaturated acylamides is reported for the first time via copper-catalyzed direct amidation between readily available cinnamic acids and N-substituted formamides. The protocol was easily accessible and practical. ... Examples of molecules containing ...

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N-Arylpiperazinyl-N'-propylamino Derivatives of Heteroaryl A...

[Elworthy, Todd R.; Ford, Anthony P. D. W.; Bantle, Gary W.; Morgans Jr., David J.; Ozer, Rachel S.; Palmer, Wylie S.; Repke, David B.; Romero, Magarita; Sandoval, Leticia; Sjogren, Eric B.; Talamas, Francisco X.; Vazquez, Alfredo; Wu, Helen; Arredondo, Nicolas F.; Blue Jr., David R.; DeSousa, Andrea; Gross, Lisa M.; Kava, M. Shannon; Lesnick, John D.; Vimont, Rachel L.; Williams, Timothy J.; Zhu, Quan-Ming; Pfister, Juerg R.; Clarke, David E. Journal of Medicinal Chemistry, 1997 , vol. 40, # 17 p. 2674 - 2687]

Studies on Organophosphorus Compounds XVI On O, O??Dialkyl D...

[Perregaard,J. et al. Bulletin des Societes Chimiques Belges, 1977 , vol. 86, p. 321 - 328]