Israel Journal of Chemistry

Nucleoside Analogues: Synthesis from Strained Rings

S Racine, J Vuilleumier, J Waser

Index: BRISTOL-MYERS SQUIBB COMPANY Patent: WO2003/99286 A1, 2003 ; Location in patent: Page 94 ;

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Citation Number: 2

Abstract

... 0000, 00, 1 – 13 0000 Wiley-VCH Verlag GmbH & Co. KGaA, Weinheim ... Page 6. ... The two-step protocol gave better yield of nucleoside ana- logues in the case of acetophenone (20): 94% yield of 23b was obtained instead of 60% of 23a without depro- tection (Scheme 7B). ...