Some heterocyclic sulfonyl chlorides and derivatives

RJ Cremlyn, FJ Swinbourne…

Index: Cremlyn, Richard J.; Swinbourne, Fred J.; Yung, Kin-Man Journal of Heterocyclic Chemistry, 1981 , vol. 18, p. 997 - 1006

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Citation Number: 17

Abstract

Abstract The syntheses of 4-and 5-chlorosulfonylfuran-2-carboxylic acid (Ia, IIa), 4- chlorosulfonylfuran-2-carboxamide (Ib), 3, 5-dimethylpyrazole and isoxazole-4-sulfonyl chlorides (IIIa, IVa) and 2, 4-dimethylthiazole-5-sulfonyl chloride (Va) are described. The sulfonyl chlorides were converted into a range of amides, hydrazides and azides. Condensation of the sulfonohydrazides with β-dicarbonyl compounds, gave the ...