Tetrahedron

Diastereoselective synthesis of 2-oxiranyl and 2-aziridinyl thiazoles

F Bona, L De Vitis, S Florio, L Ronzini, L Troisi

Index: Bona, Fabio; De Vitis, Luisella; Florio, Saverio; Ronzini, Ludovico; Troisi, Luigino Tetrahedron, 2003 , vol. 59, # 9 p. 1381 - 1387

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Citation Number: 9

Abstract

Download PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... 2-Chloroalkylthiazolyllithiums, prepared by deprotonating the 2-chloroalkylthiazoles with n-BuLi at −78°C in THF, add to ketones or imines affording in 'one-pot' oxiranes and aziridines in a Z stereoselective manner. ... The synthesis of 2-benzothiazolyl, 4 2-oxazolinyl, 5 2 (3 and ...