Synlett

Regioselective Synthesis of Substituted Imidate N-[1-Methyleneisobenzofuran-3 (1H)-ylidene] benzenamines via Palladium-Catalyzed Tandem Heteroannulation of o- …

…, X Wang, F Li, GL Gao, XM Chen, WS Wu, JJ Wang

Index: Yan, Ze-Yi; Tan, Cun-Min; Wang, Xue; Li, Fei; Gao, Guo-Lin; Chen, Xi-Meng; Wu, Wang-Suo; Wang, Jian-Jun Synlett, 2011 , # 13 p. 1863 - 1870

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Citation Number: 2

Abstract

Abstract A variety of substituted imidate N-[1-methyleneisobenzofuran-3 (1H)-ylidene] benzenamines have been prepared in good to excellent yields by the palladium-catalyzed tandem heteroannulation of o-(1-alkynyl) benzamides with iodobenzene. The products obtained from this process were unusual substituted N-[isobenzofuran-3 (1H)-ylidene] benzenamines. The tandem cyclization of readily available o-(1-alkynyl) benzamides and ...