Tetrahedron letters

Amidine derivatives of α-arylglycines from N-(1-aryl-2, 2, 2-trichloroethyl) amides of arenesulfonic acids and secondary amines

IB Rozentsveig, GG Levkovskaya, GN Rozentsveig…

Index: Rozentsveig; Levkovskaya; Mirskova Russian Journal of Organic Chemistry, 1999 , vol. 35, # 6 p. 895 - 898

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Citation Number: 26

Abstract

The interaction of N-(1-aryl-2, 2, 2-trichloroethyl) amides of arenesulfonic acids with secondary amines or their salts in the presence of inorganic bases involves the formation of chloroaziridine intermediates. Depending upon the solvent and reagent ratio, the reaction

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Synthesis and biological activity of N-(1-R-2, 2, 2-trichlor...

[Mirskova, A. N.; Drozdova, T. I.; Levkovskaya, G. G.; Kuznetsova, E. E.; Vavil'chenkova, G. S.; et al. Pharmaceutical Chemistry Journal, 1982 , vol. 16, # 12 p. 899 - 902 Khimiko-Farmatsevticheskii Zhurnal, 1982 , vol. 16, # 12 p. 1479 - 1481]