Tetrahedron letters

A fast procedure for the preparation of vicinal azidoalcohols using polymer supported reagents

ECS Brenelli, JA Brenelli, RCL Pinto

Index: Souza Brenelli, Eugenia Cristina; Brenelli, Jose Afranio; Laranjeira Pinto, Raquel Cristina Tetrahedron Letters, 2005 , vol. 46, # 27 p. 4531 - 4533

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Citation Number: 14

Abstract

Our research interests concerned the preparation of chiral 1-aryl-2-azidoethanols through biotransformations of corresponding α-azidoketones. 8 These compounds are precursors of important biologically active natural compounds. We have been using conventional solution phase chemistry to prepare racemic vicinal azidoalcohols for kinetic enzymatic resolution. 9 In order to speed up the preparation of such compounds we devised an alternative procedure using polymer supported ...