Tetrahedron Letters

Fluoroalkanosulfonyl fluorides-mediated cyclodehydration of β-hydroxy sulfonamides and β-hydroxy thioamides to the corresponding aziridines and thiazolines

Z Yan, C Guan, Z Yu, W Tian

Index: Yan, Zhaohua; Guan, Chengbo; Yu, Zhangxin; Tian, Weisheng Tetrahedron Letters, 2013 , vol. 54, # 43 p. 5788 - 5790

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Citation Number: 9

Abstract

Abstract An efficient method for the fluoroalkanosulfonyl fluoride-induced cyclodehydration of β-hydroxy sulfonamides and β-hydroxy thioamides to the corresponding aziridines and thiazolines is reported. Mild reaction conditions, operational simplicity, and high yields are the major advantages of this method.

100132-60-3

(S)-N-tosyl-alaninol

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