The Journal of Organic Chemistry

Nucleophilic Fluorination and Radiofluorination via Aziridinium Intermediates: N-Substituent Influence, Unexpected Regioselectivity, and Differences between …

M Médoc, F Sobrio

Index: Tunbridge, Gemma A.; Baruchello, Riccardo; Caggiano, Lorenzo RSC Advances, 2013 , vol. 3, # 14 p. 4613 - 4621

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Abstract

... Volume: Page: ... 12, 11, Bn, Me, 90, 14, 74, 46:54. a ... for allylic substituents compared with benzylic substituents on the amine, with a slight effect on the reaction selectivity, which is consistent with our observations using fluorine (Table 1, entries 1 and 3). In contrast ...

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