Evaluation of benzyltetrahydroisoquinolines as ligands for neuronal nicotinic acetylcholine receptors

…, E Sher, BK Cassels, I Bermudez

Index: Exley, Richard; Iturriaga-Vasquez, Patricio; Lukas, Ronald J.; Sher, Emanuele; Cassels, Bruce K.; Bermudez, Isabel British Journal of Pharmacology, 2005 , vol. 146, # 1 p. 15 - 24

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Citation Number: 13

Abstract

5 These studies suggest that C derivatives may be useful tools for studies characterising the antagonist and ion channel sites on human a7, a4b2 or a4b4 nACh receptors and for revealing structure–function relationships for nACh receptor antagonists. British Journal of Pharmacology (2005) 146, 15–24. doi: 10.1038/sj. bjp. 0706307; published online 27 June 2005 Keywords: Tetrandrine; nicotinic acetylcholine receptors; laudanosine; armepavine; ...