BMS-200475, a novel carbocyclic 2′-deoxyguanosine analog with potent and selective anti-hepatitis B virus activity in vitro

GS Bisacchi, ST Chao, C Bachard, JP Daris…

Index: Bioorganic and Medicinal Chemistry Letters, , vol. 7, # 2 p. 127 - 132

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Citation Number: 135

Abstract

... Bioorganic & Medicinal Chemistry Letters. Volume 7, Issue 2, 21 January 1997, Pages 127–132. ... A practical 10-step asymmetric synthesis was developed affording BMS-200475 in 18% overall chemical yield and >99% optical purity. ... 1. DO White, FJ Fenner; Medical Virology. ...

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