Biarylaniline phenethanolamines as potent and selective β3 adrenergic receptor agonists

DE Uehling, BG Shearer, KH Donaldson…

Index: Journal of Medicinal Chemistry, , vol. 49, # 9 p. 2758 - 2771

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Citation Number: 30

Abstract

... Journal of Medicinal ... 49 (9), pp 2758–2771. DOI: 10.1021/jm0509445. Publication Date (Web): April 13, 2006. Copyright © 2006 American Chemical Society. ... In the medicinal chemistry strategy described herein, the carboxylic acid was retained but was constrained within a biaryl ...

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Biarylaniline phenethanolamines as potent and selective β3 a...

[Uehling, David E.; Shearer, Barry G.; Donaldson, Kelly H.; Chao, Esther Y.; Deaton, David N.; Adkison, Kim K.; Brown, Kathleen K.; Cariello, Neal F.; Faison, Walter L.; Lancaster, Mary E.; Lin, Jasmine; Hart, Robert; Milliken, Tula O.; Paulik, Mark A.; Sherman, Bryan W.; Sugg, Elizabeth E.; Cowan, Conrad Journal of Medicinal Chemistry, 2006 , vol. 49, # 9 p. 2758 - 2771]

Palladium-catalyzed coupling of functionalized bromoarenes t...

[Tetrahedron Letters, , vol. 40, # 3 p. 415 - 418]