Concise Synthesis of Bicyclic Aminals by Way of Catalytic Intramolecular CH Amination and Evaluation of Their Reactivity as Iminium Precursors

D Rodríguez-Lucena, M ST Morin…

Index: Letters in Organic Chemistry, , vol. 8, # 3 p. 155 - 162

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Abstract

... 9 CH2Cl2 0°C to rt, 16 h (R = Cbz) (R = Ts) 7 R = Ts 11 DMAP 59% CH2Cl2 0°C to rt, 16 h 10 ClSO2NH2 ClSO2NH2 ClSO2NH2 Scheme 3. Page 4. 158 Letters in Organic Chemistry, 2011, Vol. 8, No. 3 Rodríguez-Lucena et al. more strained bicyclic aminal 18. ...