e.g. Filippa Pettersson or Cancer Res. 75(6) , 1102-12, (2015) or 10.1002/anie.201600521

2, 5-Disubstituted-1, 3, 4-oxadiazoles/thiadiazole as surface recognition moiety: Design and synthesis of novel hydroxamic acid based histone deacetylase inhibitors

H Rajak, A Agarawal, P Parmar, BS Thakur…

Index: Bioorganic and Medicinal Chemistry Letters, , vol. 21, # 19 p. 5735 - 5738

Full Text: HTML

Citation Number: 47

Abstract

... Bioorganic & Medicinal Chemistry Letters. ... a Medicinal Chemistry Research Laboratory, SLT Institute of ... b Chhattisgarh Institute of Medical Sciences, Bilaspur 495 009, CG, India; c Faculty of Pharmacy, AIMST University, Semeling, Bedong 08100, Kedah Darul Aman, Malaysia; ...

4-Chlorobenzaldehyde Structure

4-Chlorobenzaldehyde

~%

5-(4-chlorophenyl)-1,3,4-thiadiazol-2-amine Structure

5-(4-chlorophen...

4-Methoxybenzaldehyde Structure

4-Methoxybenzal...

~%

2-AMINO-5-(4-METHOXYPHENYL)-1,3,4-OXADIAZOLE Structure

2-AMINO-5-(4-ME...

4-Methoxybenzaldehyde Structure

4-Methoxybenzal...

~%

2-Amino-5-(4-methoxyphenyl)-1,3,4-thiadiazole Structure

2-Amino-5-(4-me...

2-Chlorobenzaldehyde Structure

2-Chlorobenzaldehyde

~%

2-Amino-5-(2-chlorophenyl)-1,3,4-oxadiazole Structure

2-Amino-5-(2-ch...

p-Nitrobenzaldehyde thiosemicarbazone Structure

p-Nitrobenzalde...

~77%

1,3,4-Thiadiazol-2-amine,5-(4-nitrophenyl)- Structure

1,3,4-Thiadiazo...

4-Nitrobenzaldehyde Structure

4-Nitrobenzaldehyde

~%

1,3,4-Thiadiazol-2-amine,5-(4-nitrophenyl)- Structure

1,3,4-Thiadiazo...

4-Fluorobenzaldehyde Structure

4-Fluorobenzaldehyde

~%

5-(4-Fluorophenyl)-1,3,4-oxadiazol-2-amine Structure

5-(4-Fluorophen...

Benzaldehyde Structure

~%

5-Phenyl-1,3,4-thiadiazol-2-amine Structure

5-Phenyl-1,3,4-...

3-Chlorobenzaldehyde Structure

3-Chlorobenzaldehyde

~%

5-(3-Chlorophenyl)-1,3,4-oxadiazol-2-amine Structure

5-(3-Chlorophen...

Synthesis of 2-N-salicylidene-5-(substituted)-1, 3, 4-thiadi...

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A convenient and general synthesis of 2??amino??1, 3, 4??thi...

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FeCl3-promoted synthesis of 1, 3, 4-thiadiazoles under combi...

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Recherche de paramètres structuraux influençant l'activité a...

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Efficient synthesis of antifungal active 9-substituted-3-ary...

[Bioorganic and Medicinal Chemistry Letters, , vol. 21, # 16 p. 4919 - 4923]